Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

Chelliah Selvam; Isabelle A. Lemasson; Isabelle Brabet; Nadia Oueslati; Berin Karaman; Alexandre Cabaye; Amélie S. Tora; Bruno Commare; Tiphanie Courtiol; Sara Cesarini; Isabelle McCort-Tranchepain; Delphine Rigault; Laetitia Mony; Thomas Bessiron; Heather McLean; Frédéric R. Leroux; Françoise Colobert; Hervé Daniel; Anne Goupil-Lamy; Hugues Olivier Bertrand; Cyril Goudet; Jean Philippe Pin; Francine C. Acher

doi:10.1021/acs.jmedchem.7b01438

Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

Chelliah Selvam, Isabelle A. Lemasson, Isabelle Brabet, Nadia Oueslati, Berin Karaman, Alexandre Cabaye, Amélie S. Tora, Bruno Commare, Tiphanie Courtiol, Sara Cesarini, Isabelle McCort-Tranchepain, Delphine Rigault, Laetitia Mony, Thomas Bessiron, Heather McLean, Frédéric R. Leroux, Françoise Colobert, Hervé Daniel, Anne Goupil-Lamy, Hugues Olivier BertrandCyril Goudet, Jean Philippe Pin, Francine C. Acher

Texas Southern University

Research output: Contribution to journal › Article › peer-review

Original language	English
Pages (from-to)	1969-1989
Number of pages	21
Journal	Journal of Medicinal Chemistry
Volume	61
Issue number	5
DOIs	https://doi.org/10.1021/acs.jmedchem.7b01438
State	Published - Mar 8 2018

ASJC Scopus Subject Areas

Molecular Medicine
Drug Discovery

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10.1021/acs.jmedchem.7b01438

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Selvam, C., Lemasson, I. A., Brabet, I., Oueslati, N., Karaman, B., Cabaye, A., Tora, A. S., Commare, B., Courtiol, T., Cesarini, S., McCort-Tranchepain, I., Rigault, D., Mony, L., Bessiron, T., McLean, H., Leroux, F. R., Colobert, F., Daniel, H., Goupil-Lamy, A., ... Acher, F. C. (2018). Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. Journal of Medicinal Chemistry, 61(5), 1969-1989. https://doi.org/10.1021/acs.jmedchem.7b01438

Selvam, C, Lemasson, IA, Brabet, I, Oueslati, N, Karaman, B, Cabaye, A, Tora, AS, Commare, B, Courtiol, T, Cesarini, S, McCort-Tranchepain, I, Rigault, D, Mony, L, Bessiron, T, McLean, H, Leroux, FR, Colobert, F, Daniel, H, Goupil-Lamy, A, Bertrand, HO, Goudet, C, Pin, JP & Acher, FC 2018, 'Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites', Journal of Medicinal Chemistry, vol. 61, no. 5, pp. 1969-1989. https://doi.org/10.1021/acs.jmedchem.7b01438

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doi = "10.1021/acs.jmedchem.7b01438",

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AU - Selvam, Chelliah

AU - Lemasson, Isabelle A.

AU - Brabet, Isabelle

AU - Oueslati, Nadia

AU - Karaman, Berin

AU - Cabaye, Alexandre

AU - Tora, Amélie S.

AU - Commare, Bruno

AU - Courtiol, Tiphanie

AU - Cesarini, Sara

AU - McCort-Tranchepain, Isabelle

AU - Rigault, Delphine

AU - Mony, Laetitia

AU - Bessiron, Thomas

AU - McLean, Heather

AU - Leroux, Frédéric R.

AU - Colobert, Françoise

AU - Daniel, Hervé

AU - Goupil-Lamy, Anne

AU - Bertrand, Hugues Olivier

AU - Goudet, Cyril

AU - Pin, Jean Philippe

AU - Acher, Francine C.

PY - 2018/3/8

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JO - Journal of Medicinal Chemistry

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IS - 5

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Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

ASJC Scopus Subject Areas

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