Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

Chelliah Selvam; Isabelle A. Lemasson; Isabelle Brabet; Nadia Oueslati; Berin Karaman; Alexandre Cabaye; Amélie S. Tora; Bruno Commare; Tiphanie Courtiol; Sara Cesarini; Isabelle McCort-Tranchepain; Delphine Rigault; Laetitia Mony; Thomas Bessiron; Heather McLean; Frédéric R. Leroux; Françoise Colobert; Hervé Daniel; Anne Goupil-Lamy; Hugues Olivier Bertrand; Cyril Goudet; Jean Philippe Pin; Francine C. Acher

doi:10.1021/acs.jmedchem.7b01438

Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

Chelliah Selvam
, Isabelle A. Lemasson
, Isabelle Brabet
, Nadia Oueslati
, Berin Karaman
, Alexandre Cabaye
, Amélie S. Tora
, Bruno Commare
, Tiphanie Courtiol
, Sara Cesarini
, Isabelle McCort-Tranchepain
, Delphine Rigault
, Laetitia Mony
, Thomas Bessiron
, Heather McLean
, Frédéric R. Leroux
, Françoise Colobert
, Hervé Daniel
, Anne Goupil-Lamy
, Hugues Olivier Bertrand

Cyril Goudet, Jean Philippe Pin, Francine C. Acher

Texas Southern University

Research output: Contribution to journal › Article › peer-review

Original language	English
Pages (from-to)	1969-1989
Number of pages	21
Journal	Journal of Medicinal Chemistry
Volume	61
Issue number	5
DOIs	https://doi.org/10.1021/acs.jmedchem.7b01438
State	Published - Mar 8 2018

ASJC Scopus Subject Areas

Molecular Medicine
Drug Discovery

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10.1021/acs.jmedchem.7b01438

Cite this

Selvam, C., Lemasson, I. A., Brabet, I., Oueslati, N., Karaman, B., Cabaye, A., Tora, A. S., Commare, B., Courtiol, T., Cesarini, S., McCort-Tranchepain, I., Rigault, D., Mony, L., Bessiron, T., McLean, H., Leroux, F. R., Colobert, F., Daniel, H., Goupil-Lamy, A., ... Acher, F. C. (2018). Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. Journal of Medicinal Chemistry, 61(5), 1969-1989. https://doi.org/10.1021/acs.jmedchem.7b01438

Selvam, C, Lemasson, IA, Brabet, I, Oueslati, N, Karaman, B, Cabaye, A, Tora, AS, Commare, B, Courtiol, T, Cesarini, S, McCort-Tranchepain, I, Rigault, D, Mony, L, Bessiron, T, McLean, H, Leroux, FR, Colobert, F, Daniel, H, Goupil-Lamy, A, Bertrand, HO, Goudet, C, Pin, JP & Acher, FC 2018, 'Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites', Journal of Medicinal Chemistry, vol. 61, no. 5, pp. 1969-1989. https://doi.org/10.1021/acs.jmedchem.7b01438

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author = "Chelliah Selvam and Lemasson, \{Isabelle A.\} and Isabelle Brabet and Nadia Oueslati and Berin Karaman and Alexandre Cabaye and Tora, \{Am{\'e}lie S.\} and Bruno Commare and Tiphanie Courtiol and Sara Cesarini and Isabelle McCort-Tranchepain and Delphine Rigault and Laetitia Mony and Thomas Bessiron and Heather McLean and Leroux, \{Fr{\'e}d{\'e}ric R.\} and Fran{\c c}oise Colobert and Herv{\'e} Daniel and Anne Goupil-Lamy and Bertrand, \{Hugues Olivier\} and Cyril Goudet and Pin, \{Jean Philippe\} and Acher, \{Francine C.\}",

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doi = "10.1021/acs.jmedchem.7b01438",

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AU - Selvam, Chelliah

AU - Lemasson, Isabelle A.

AU - Brabet, Isabelle

AU - Oueslati, Nadia

AU - Karaman, Berin

AU - Cabaye, Alexandre

AU - Tora, Amélie S.

AU - Commare, Bruno

AU - Courtiol, Tiphanie

AU - Cesarini, Sara

AU - McCort-Tranchepain, Isabelle

AU - Rigault, Delphine

AU - Mony, Laetitia

AU - Bessiron, Thomas

AU - McLean, Heather

AU - Leroux, Frédéric R.

AU - Colobert, Françoise

AU - Daniel, Hervé

AU - Goupil-Lamy, Anne

AU - Bertrand, Hugues Olivier

AU - Goudet, Cyril

AU - Pin, Jean Philippe

AU - Acher, Francine C.

PY - 2018/3/8

Y1 - 2018/3/8

UR - https://www.scopus.com/pages/publications/85043467137

UR - https://www.scopus.com/pages/publications/85043467137#tab=citedBy

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C2 - 29397723

AN - SCOPUS:85043467137

SN - 0022-2623

VL - 61

SP - 1969

EP - 1989

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

IS - 5

ER -

Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites

ASJC Scopus Subject Areas

Access to Document

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